NO140057C - ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE ALFA-ARYL-4-SUBSTITUTED PIPERIDINOAL CANOL DERIVATIVES - Google Patents

ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE ALFA-ARYL-4-SUBSTITUTED PIPERIDINOAL CANOL DERIVATIVES

Info

Publication number: NO140057C
Authority: NO; Norway
Prior art keywords: piperidinoal; canol; aryl; derivatives; substituted
Prior art date: 1972-01-28

Application number

NO326/73A

Other languages

Norwegian (no)

Other versions

NO140057B (en

Inventor

Albert Anthony Carr

Clyde Richard Kinsolving

Original Assignee

Richardson Merrell Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1972-01-28

Filing date

1973-01-26

Publication date

1979-07-04

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22829539&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO140057(C) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1973-01-26 Application filed by Richardson Merrell Inc filed Critical Richardson Merrell Inc

1979-03-19 Publication of NO140057B publication Critical patent/NO140057B/en

1979-07-04 Publication of NO140057C publication Critical patent/NO140057C/en

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D211/70—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/10—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms
- C07D211/14—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms with hydrocarbon or substituted hydrocarbon radicals attached to the ring nitrogen atom
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D211/20—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
- C07D211/22—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms by oxygen atoms

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Hydrogenated Pyridines (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

NO326/73A 1972-01-28 1973-01-26 ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE ALFA-ARYL-4-SUBSTITUTED PIPERIDINOAL CANOL DERIVATIVES NO140057C (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US22182172A	1972-01-28	1972-01-28

Publications (2)

Publication Number	Publication Date
NO140057B NO140057B (en)	1979-03-19
NO140057C true NO140057C (en)	1979-07-04

Family

ID=22829539

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO326/73A NO140057C (en)	1972-01-28	1973-01-26	ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE ALFA-ARYL-4-SUBSTITUTED PIPERIDINOAL CANOL DERIVATIVES

Country Status (26)

Country	Link
JP (1)	JPS5115035B2 (en)
AR (1)	AR195314A1 (en)
AT (2)	AT321917B (en)
AU (1)	AU467361B2 (en)
BE (1)	BE794597A (en)
CA (1)	CA978946A (en)
CH (2)	CH593259A5 (en)
CS (1)	CS177834B2 (en)
DD (1)	DD103239A5 (en)
DE (1)	DE2303306C3 (en)
DK (1)	DK136713B (en)
ES (1)	ES410731A1 (en)
FR (1)	FR2181690B1 (en)
GB (1)	GB1413138A (en)
HU (1)	HU166477B (en)
IE (1)	IE36983B1 (en)
IL (1)	IL41060A (en)
LU (1)	LU66916A1 (en)
NL (1)	NL175410C (en)
NO (1)	NO140057C (en)
PH (1)	PH10264A (en)
PL (1)	PL89095B1 (en)
SE (1)	SE382058B (en)
SU (1)	SU464997A3 (en)
YU (1)	YU36013B (en)
ZA (1)	ZA728544B (en)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3941795A (en)	1974-02-08	1976-03-02	Richardson-Merrell Inc.	α-ARYL-4-SUBSTITUTED PIPERIDINOALKANOL DERIVATIVES
US4254130A (en) *	1979-04-10	1981-03-03	Richardson-Merrell Inc.	Piperidine derivatives
US4254129A (en) *	1979-04-10	1981-03-03	Richardson-Merrell Inc.	Piperidine derivatives
IT1200123B (en) *	1985-09-27	1989-01-05	Ind Chimica Srl	PROCESS FOR ALPHA PREPARATION
US4742175A (en) *	1986-05-07	1988-05-03	Merrell Dow Pharmaceuticals Inc.	Preparation of polymorphically pure terfenadine
JPS63101760U (en) *	1986-12-19	1988-07-02
IT1205685B (en) *	1987-05-26	1989-03-31	Erregierre Spa	PROCESS FOR THE PREPARATION OF ALPHA- (ALCHYLPHENYL) -4- (HYDROXY DIPHENYLMETHYL) -1-PIPERIDINE BUTANOL
IL93499A0 (en) *	1989-02-28	1990-11-29	Merrell Dow Pharma	Preparation of the low melting polymorphic form of terfenadine
CA2015390A1 (en) *	1989-05-01	1990-11-01	Frederick J. Mccarty	Process for the preparation of the high melting polymorphic of terfenadine
DE3917241A1 (en) *	1989-05-26	1990-11-29	Schaper & Bruemmer Gmbh	4- (HYDROXYDIPHENYLMETHYL) -1-PIPERIDYL-PHENYLALKANE DERIVATIVES
US5466691A (en) *	1991-08-09	1995-11-14	Yoshitomi Pharmaceutical Industries, Ltd.	Thiophene compound
CA2216877A1 (en) *	1995-05-08	1996-11-14	Hoechst Marion Roussel, Inc.	Alpha-(substituted alkylphenyl)-4-(hydroxydiphenylmethyl)-1-piperidine butanol derivatives, their preparation and their use as anti-histamines, anti-allergy agents and bronchodilators
ES2216191T3 (en) *	1997-03-11	2004-10-16	Aventis Pharmaceuticals Inc.	PROCEDURE FOR PREPARING ACID 4- (4- (HYDROXIDIFENYL) -1-PIPERIDINYL) -1-HYDROXIBUTE) -ALFA, ALPHA-DIMETHYLPHENYLACETIC AND PHOSPHORILE DERIVATIVES.
US7498345B2 (en) *	2004-09-17	2009-03-03	Albany Molecular Research, Inc.	Process for production of piperidine derivatives
US8153385B2 (en)	2004-10-18	2012-04-10	Reverse Proteomics Research Institute Co., Ltd.	Target protein and target gene in drug designing and screening method

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3081303A (en) *	1961-10-13	1963-03-12	Searle & Co	1-aminoalkyl-alpha, alpha-diphenylpiperidine-methanols
GB1242169A (en) *	1969-04-09	1971-08-11	Ucb Sa	Piperidine derivatives

1972
- 1972-12-04 ZA ZA728544A patent/ZA728544B/en unknown
- 1972-12-05 IE IE1689/72A patent/IE36983B1/en unknown
- 1972-12-08 PH PH14156A patent/PH10264A/en unknown
- 1972-12-11 AU AU49893/72A patent/AU467361B2/en not_active Ceased
- 1972-12-12 IL IL41060A patent/IL41060A/en unknown
- 1972-12-15 GB GB5799572A patent/GB1413138A/en not_active Expired
- 1972-12-20 CH CH1381476A patent/CH593259A5/xx not_active IP Right Cessation
- 1972-12-20 CH CH1854272A patent/CH587820A5/xx not_active IP Right Cessation
- 1972-12-27 JP JP47130136A patent/JPS5115035B2/ja not_active Expired
- 1972-12-29 AT AT1115372A patent/AT321917B/en not_active IP Right Cessation
- 1972-12-29 AT AT246074*1A patent/AT323742B/en not_active IP Right Cessation
1973
- 1973-01-08 YU YU34/73A patent/YU36013B/en unknown
- 1973-01-16 CA CA161,413A patent/CA978946A/en not_active Expired
- 1973-01-17 HU HURI498A patent/HU166477B/hu unknown
- 1973-01-18 ES ES410731A patent/ES410731A1/en not_active Expired
- 1973-01-22 NL NLAANVRAGE7300873,A patent/NL175410C/en not_active IP Right Cessation
- 1973-01-24 FR FR7302503A patent/FR2181690B1/fr not_active Expired
- 1973-01-24 DE DE2303306A patent/DE2303306C3/en not_active Expired
- 1973-01-24 SE SE7300974A patent/SE382058B/en active Protection Beyond IP Right Term
- 1973-01-25 DD DD168482A patent/DD103239A5/xx unknown
- 1973-01-26 CS CS630A patent/CS177834B2/cs unknown
- 1973-01-26 BE BE794597D patent/BE794597A/en not_active IP Right Cessation
- 1973-01-26 PL PL1973160419A patent/PL89095B1/pl unknown
- 1973-01-26 LU LU66916A patent/LU66916A1/xx unknown
- 1973-01-26 DK DK44973AA patent/DK136713B/en not_active IP Right Cessation
- 1973-01-26 AR AR246313A patent/AR195314A1/en active
- 1973-01-26 NO NO326/73A patent/NO140057C/en unknown
- 1973-01-27 SU SU1878074A patent/SU464997A3/en active

Also Published As

Publication number	Publication date
NL7300873A (en)	1973-07-31
YU3473A (en)	1981-02-28
CH593259A5 (en)	1977-11-30
PL89095B1 (en)	1976-10-30
IL41060A (en)	1975-06-25
FR2181690B1 (en)	1976-05-14
IE36983B1 (en)	1977-04-13
ES410731A1 (en)	1976-04-01
DD103239A5 (en)	1974-01-12
HU166477B (en)	1975-03-28
LU66916A1 (en)	1973-07-27
AR195314A1 (en)	1973-09-28
DK136713B (en)	1977-11-14
AU467361B2 (en)	1975-11-27
NL175410B (en)	1984-06-01
FR2181690A1 (en)	1973-12-07
NL175410C (en)	1984-11-01
CS177834B2 (en)	1977-08-31
JPS5115035B2 (en)	1976-05-13
DE2303306B2 (en)	1978-09-28
NO140057B (en)	1979-03-19
BE794597A (en)	1973-05-16
IE36983L (en)	1973-07-28
IL41060A0 (en)	1973-02-28
AT321917B (en)	1975-04-25
CA978946A (en)	1975-12-02
DE2303306C3 (en)	1979-05-31
AU4989372A (en)	1974-06-13
PH10264A (en)	1976-10-20
SU464997A3 (en)	1975-03-25
YU36013B (en)	1981-11-13
SE382058B (en)	1976-01-12
ZA728544B (en)	1974-02-27
DK136713C (en)	1978-05-01
GB1413138A (en)	1975-11-05
DE2303306A1 (en)	1973-08-02
CH587820A5 (en)	1977-05-13
AT323742B (en)	1975-07-25
JPS4885578A (en)	1973-11-13

Publication	Publication Date	Title
NO140059C (en)	1979-07-04	ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE SUBSTITUTED PIPERIDINE DERIVATIVES
NO793013L (en)	1973-11-06	ANALOGICAL PROCEDURES FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE BENZODIAZEPIN DERIVATIVES
NO139560C (en)	1979-04-04	ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY EFFECTIVE NONAPEPTIDAMIDE DERIVATIVES
NO137941C (en)	1978-05-31	ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE TRI-P-TOLUENESULPHONATE OF S-ADENOSYL-L-METHIONINE
NO140381C (en)	1979-08-22	ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE ARYLPIPERAZINES
NO138565C (en)	1978-09-27	ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE PIPERAZINYL-PROPYL-1,2,4-TRIAZOLINON DERIVATIVES
NO140058C (en)	1979-07-04	ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE SUBSTITUTED PIPERIDINOALCANOL-OXIM DERIVATIVES
NO136094C (en)	1977-07-20	ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE D-1- (4-AMINO-PHENYL) -2-ALKYLAMINO-ETHANOL DERIVATIVES.
NO149281C (en)	1984-03-21	ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE 7ALFA METHOXYPHALOSPORINE DERIVATIVES
NO140057C (en)	1979-07-04	ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE ALFA-ARYL-4-SUBSTITUTED PIPERIDINOAL CANOL DERIVATIVES
NO138999C (en)	1978-12-20	ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE DIPHENYLYL-ALKANOYLAMINOPYRIDINES
NO140597C (en)	1979-10-03	ANALOGICAL PROCEDURES FOR THE PREPARATION OF THERAPEUTIC ACTIVE 8-AZAPURIN-6-ON DERIVATIVES
NO140670C (en)	1979-10-17	ANALOGICAL PROCEDURES FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE PYRAZOLODIAZEPIN DERIVATIVES
NO140821C (en)	1979-11-21	ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE PYRIDO-PYRIMIDINE DERIVATIVES
NO137858C (en)	1978-05-10	ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE INDANONS
NO142260C (en)	1980-07-23	ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE TIENOTRIAZOLODIAZEPINE DERIVATIVES
NO138063C (en)	1978-06-21	ANALOGICAL PROCEDURE FOR PREPARATION OF THERAPEUTICALLY ACTIVE NORMORPHINON DERIVATIVES
NO137728C (en)	1978-04-12	ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE PYRASI-4-OXYDE DERIVATIVES
NO143499C (en)	1981-02-25	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE INHANDER DERIVATIVES
NO140299C (en)	1979-08-08	ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE 4-ARYL-5-AMINOALKYL-4-OXSAZOLIN-2-ONERS
NO138251C (en)	1978-08-02	ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE BENZYLAMINES
NO139050C (en)	1979-01-03	ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE NORORIPAVIN AND TEBAIN DERIVATIVES
NO138285C (en)	1978-08-09	ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE LINCOMYCIN DERIVATIVES
NO137695C (en)	1978-04-05	ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE N-THENYLMETHYL-HETEROCYCLIC COMPOUNDS
NO137727C (en)	1978-04-12	ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE 1-PHENYL-3-HYDROXY-3-METHYLTRIAZENES